Design, synthesis and biological evaluation of second-generation benzoylpiperidine derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
Carlotta Granchi, Giulia Bononi, Rebecca Ferrisi, Eleonora Gori, Giulia Mantini, Sandra Glasmacher, Giulio Poli, Stefano Palazzolo, Isabella Caligiuri, Flavio Rizzolio, Vincenzo Canzonieri, Tiziana Perin, Jürg Gertsch, Andrea Sodi, Elisa Giovannetti, Marco Macchia, Filippo Minutolo, Tiziano Tuccinardi, Andrea Chicca
Topics & Concepts
Monoacylglycerol lipaseEndocannabinoid systemChemistryEnzymeBiochemistryPharmacologyCancer researchBiologyReceptorCannabis and Cannabinoid ResearchPancreatic function and diabetesDiet, Metabolism, and Disease