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Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment

Adel A. Marzouk, Ehab S. Taher, Montaser Sh. A. Shaykoon, Ping Lan, Walaa Hamada Abd‐Allah, Adel Mohamed Aboregela, Mohammed Farrag El‐Behairy

2021Bioorganic Chemistry24 citationsDOI

Topics & Concepts

In vivoChemistryPharmacologyCelecoxibApoptosisPyrazoleEdemaIn vitroSelectivityGene expressionBiochemistryGeneStereochemistryBiologyInternal medicineMedicineBiotechnologyCatalysisSynthesis and biological activityInflammatory mediators and NSAID effectsComputational Drug Discovery Methods
Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment | Litcius