Synthesis, biological evaluation and molecular docking studies of new pyrimidine derivatives as potent dual EGFR/HDAC inhibitors
G. Sivaiah, M.S. Raghu, S. Prasad, A.M. Anusuya, K. Yogesh Kumar, Fahd Alharethy, M.K. Prashanth, Byong‐Hun Jeon
Topics & Concepts
ChemistryDocking (animal)EGFR inhibitorsVorinostatPharmacophorePyrimidineEpidermal growth factor receptorHistone deacetylaseErlotinibHDAC1HDAC6A549 cellBiochemistryIC50PharmacologyIn vitroCombinatorial chemistryHistoneReceptorMedicineNursingGeneHistone Deacetylase Inhibitors ResearchBiochemical and Molecular ResearchQuinazolinone synthesis and applications