Litcius/Paper detail

A two-metalloenzyme cascade constructs the azetidine-containing pharmacophore

Rong Gong, Yao Qu, Jia Liu, Xuan Zhang, Liwei Zhou, Tian Zhu, Xinyue Zeng, Bo Jin, Zhen Li, Le Yu, Ruyi Chen, Yang Zhou, Langxing Liao, Liulin Yang, Xuemin Song, You‐Sheng Cai, Kun Shen, Zixin Deng, Zhengyu Zhang, Binju Wang, Wenqing Chen

2025Nature Chemistry9 citationsDOI

Topics & Concepts

ChemistryPharmacophoreMoietyIntramolecular forceStereochemistryCascadeCombinatorial chemistryRational designEnzymeMechanism (biology)Dual (grammatical number)Dual roleDrug discoveryMoleculeSmall moleculeStereoisomerismAzetidinePhthalimideCascade reactionMolecular conformationSynthesis and Catalytic ReactionsCyclopropane Reaction MechanismsChemical Synthesis and Analysis