Design, synthesis and biological evaluation of purine-based derivatives as novel JAK2/BRD4(BD2) dual target inhibitors
Yong Guo, Yurong Zou, Yong Chen, Dexin Deng, Zihao Zhang, Kongjun Liu, Minghai Tang, Tao Yang, Suhong Fu, Chufeng Zhang, Wenting Si, Ziyan Ma, Shunjie Zhang, Bin Peng, Dingguo Xu, Lijuan Chen, Lijuan Chen
Topics & Concepts
ChemistryPharmacologyPotencyJanus kinase 2KinaseJanus kinaseIC50In vitroCancer researchBiochemistryMedicineProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsImmune Cell Function and Interaction