1,2,4-Triazolo[1,5-a]pyrimidines: Efficient one-step synthesis and functionalization as influenza polymerase PA-PB1 interaction disruptors
Maria Chiara Pismataro, Tommaso Felicetti, Chiara Bertagnin, Maria Giulia Nizi, Anna Bonomini, Maria Letizia Barreca, Violetta Cecchetti, Dirk Jochmans, Steven De Jonghe, Johan Neyts, Arianna Loregian, Oriana Tabarrini, Serena Massari
Topics & Concepts
ChemistryMoietyPyrimidineStereochemistryRNA polymeraseCombinatorial chemistryPolymeraseEC50IC50Influenza A virusIn vitroRNAEnzymeOrganic chemistryBiochemistryVirusGeneVirologyBiologyInfluenza Virus Research StudiesRespiratory viral infections researchinterferon and immune responses