Litcius/Paper detail

1,2,4-Triazolo[1,5-a]pyrimidines: Efficient one-step synthesis and functionalization as influenza polymerase PA-PB1 interaction disruptors

Maria Chiara Pismataro, Tommaso Felicetti, Chiara Bertagnin, Maria Giulia Nizi, Anna Bonomini, Maria Letizia Barreca, Violetta Cecchetti, Dirk Jochmans, Steven De Jonghe, Johan Neyts, Arianna Loregian, Oriana Tabarrini, Serena Massari

2021European Journal of Medicinal Chemistry33 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryMoietyPyrimidineStereochemistryRNA polymeraseCombinatorial chemistryPolymeraseEC50IC50Influenza A virusIn vitroRNAEnzymeOrganic chemistryBiochemistryVirusGeneVirologyBiologyInfluenza Virus Research StudiesRespiratory viral infections researchinterferon and immune responses