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Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold

Giulia Bononi, Giacomo Tonarini, Giulio Poli, Ivana Barravecchia, Isabella Caligiuri, Marco Macchia, Flavio Rizzolio, Gian Carlo Demontis, Filippo Minutolo, Carlotta Granchi, Tiziano Tuccinardi

2021European Journal of Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

Monoacylglycerol lipaseEndocannabinoid systemChemistryEnzymeContext (archaeology)Diacylglycerol lipaseLipaseBiochemistryPharmacologyBiologyPaleontologyReceptorCannabis and Cannabinoid ResearchPharmacological Receptor Mechanisms and EffectsForensic Toxicology and Drug Analysis
Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold | Litcius