Litcius/Paper detail

Tacrine – Benzothiazoles: Novel class of potential multitarget anti-Alzheimeŕs drugs dealing with cholinergic, amyloid and mitochondrial systems

Eugenie Nepovimová, Lucie Svobodová, Rafael Doležal, Vendula Hepnarová, Lucie Junova, Daniel Jun, Jan Korábečný, Tomáš Kučera, Zuzana Gažová, Katarina Motykova, Jana Kubačková, Zuzana Bednáriková, Jana Janočková, Catarina S. H. Jesus, Luísa Cortes, João Pina, Danijela Rostohar, Carlos Serpa, Ondřej Soukup, Laura Aitken, Rebecca E. Hughes, Kamil Musílek, Ľubica Múčková, Petr Jošt, Markéta Chvojková, Karel Valeš, Martin Vališ, Žofia Chrienová, Katarina Chalupova, Kamil Kuča

2020Bioorganic Chemistry32 citationsDOI

Topics & Concepts

TacrineBenzothiazoleChemistryAcetylcholinesteraseIn vivoCholinergicPharmacologyAchéIn vitroAmyloid (mycology)AmnesiaBiophysicsStereochemistryBiochemistryEnzymeNeuroscienceBiologyPsychologyBiotechnologyPsychiatryInorganic chemistryCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments