Covalent allosteric modulation: An emerging strategy for GPCRs drug discovery
Yuemin Bian, Jaden Jungho Jun, Jacob Cuyler, Xiang‐Qun Xie
Topics & Concepts
Allosteric regulationChemistryG protein-coupled receptorDrug discoveryAllosteric modulatorCovalent bondAllosteric enzymeBiochemistryReceptorOrganic chemistryReceptor Mechanisms and SignalingChemical Synthesis and AnalysisMonoclonal and Polyclonal Antibodies Research