Discovery of 5-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)-1H-indole-2-carboxamide derivatives as novel anti-cancer agents targeting Nur77
Jingbo Qin, Xiaohui Chen, Weihao Liu, Jun Chen, Weirong Liu, Yongzhen Xia, Zhehui Li, Mingyu Li, Shaojuan Wang, Quan Yuan, Ying‐Kun Qiu, Zhenhua Wu, Meijuan Fang
Topics & Concepts
ChemistryNerve growth factor IBCelastrolCancer cellCarboxamideIn vivoLead compoundApoptosisCancerStereochemistryCancer researchPharmacologyIn vitroBiochemistryNuclear receptorTranscription factorBiologyMedicineInternal medicineBiotechnologyGeneNuclear Receptors and SignalingSynthesis of Tetrazole DerivativesMacrophage Migration Inhibitory Factor