Targeted methylation facilitates DNA double strand breaks and enhances cancer suppression: A DNA intercalating/methylating dual-action chimera Amonafidazene
Dipak Walunj, Ebaston Thankarajan, Chandrashekhar Prasad, Helena Tuchinsky, Simone Baldan, Michael Y. Sherman, L. D. Patsenker, Gary Gellerman
Topics & Concepts
ChemistryChimera (genetics)DNACancer cellDNA damageMolecular biologyBiochemistryCancer researchCancerBiologyGeneticsGeneCancer therapeutics and mechanismsLung Cancer Research StudiesSynthesis and Biological Evaluation