Antibody-Based Receptor Targeting Using an Fc-Binding Peptide-Dodecaborate Conjugate and Macropinocytosis Induction for Boron Neutron Capture Therapy
Ikuhiko Nakase, Ayako Aoki, Yuriko Ito Sakai, Shiori Hirase, Miki Ishimura, Tomoka Takatani‐Nakase, Yoshihide Hattori, Mitsunori Kirihata
Abstract
assay that macropinocytosis induction during antibody-based drug delivery is crucial for the biological activity of BNCT.
Topics & Concepts
Cancer researchConjugateAntibodyCancerNeutron captureCancer cellChemistryBoronMedicineImmunologyInternal medicineMathematical analysisMathematicsOrganic chemistryBoron Compounds in ChemistryBoron and Carbon Nanomaterials ResearchRadiopharmaceutical Chemistry and Applications