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Integrating artificial intelligence into small molecule development for precision cancer immunomodulation therapy

Henry Sutanto, Deasy Fetarayani

2025npj Drug Discovery.14 citationsDOIOpen Access PDF

Abstract

This perspective examines how artificial intelligence (AI) is transforming small-molecule development for precision cancer immunomodulation therapy. It outlines AI-driven approaches for de novo design, virtual screening, multi-parameter optimization, and ADMET prediction, targeting immune checkpoints, tumor microenvironment modulation, antigen presentation, and metabolic pathways. The article highlights patient stratification, multi-omics integration, digital twin simulations, translational challenges, and future directions, underscoring AI’s potential to deliver effective, personalized immunomodulatory therapeutics.

Topics & Concepts

Immune systemPrecision medicineComputational biologyCancerTumor microenvironmentSmall moleculeComputer scienceMedicinePerspective (graphical)Personalized medicineImmunotherapyBioinformaticsCancer immunotherapyTranslational researchCancer therapyArtificial intelligenceApplications of artificial intelligenceAntigenBiologyCancer researchCancer treatmentImmunologyNeuroscienceCell Image Analysis TechniquesComputational Drug Discovery MethodsCancer Research and Treatments
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