Physiologically based pharmacokinetic modeling and simulation to predict drug–drug interactions of ivosidenib with CYP3A perpetrators in patients with acute myeloid leukemia
Chandra Prakash, Bin Fan, Alice Ke, Kha Le, Hua Yang
Topics & Concepts
CmaxCYP3A4PharmacokineticsCminItraconazolePharmacologyPhysiologically based pharmacokinetic modellingCYP3AMedicineKetoconazoleDrug-drug interactionMyeloid leukemiaInternal medicineAntifungalCytochrome P450DermatologyMetabolismChronic Myeloid Leukemia TreatmentsAcute Myeloid Leukemia ResearchMultiple Myeloma Research and Treatments