Litcius/Paper detail

Synthesis, biological evaluation and modeling of hybrids from tetrahydro-1H-pyrazolo[3,4-b]quinolines as dual cholinestrase and COX-2 inhibitors

Mohamed Mroueh, Wissam H. Faour, Wassim N. Shebaby, Costantine F. Daher, Tamer M. Ibrahim, Hanan M. Ragab

2020Bioorganic Chemistry37 citationsDOI

Topics & Concepts

ChemistryTacrineIn silicoCelecoxibIn vivoIn vitroDocking (animal)CyclooxygenaseNeuroinflammationPharmacologyEnzymeAcetylcholinesteraseBiochemistryInflammationImmunologyGeneNursingMedicineBiotechnologyBiologyCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity
Synthesis, biological evaluation and modeling of hybrids from tetrahydro-1H-pyrazolo[3,4-b]quinolines as dual cholinestrase and COX-2 inhibitors | Litcius