Design, synthesis and<i>in vitro</i>antiproliferative activity of new thiazolidinedione-1,3,4-oxadiazole hybrids as thymidylate synthase inhibitors
Zohor Mohammad Mahdi Alzhrani, Mohammad Mahboob Alam, Thikryat Neamatallah, Syed Nazreen
Abstract
has the potential to be developed as TS inhibitors.
Topics & Concepts
Thymidylate synthaseChemistryOxadiazoleCytotoxicityIn vitroIC50Cell cultureEnzymeStereochemistryDocking (animal)BiochemistryBiologyMedicineOrganic chemistryFluorouracilGeneticsChemotherapyNursingBiochemical and Molecular ResearchColorectal Cancer Treatments and StudiesSynthesis and biological activity