Pristine 2-chloroquinoline-based-thiosemicarbazones as multitarget agents against alzheimer's disease: In vitro and in silico studies of monoamine oxidase (MAO) and cholinesterase (ChE) inhibitors
Saquib Jalil, Rabia Basri, Mubashir Aziz, Zahid Shafiq, Syeda Abida Ejaz, Abdul Hameed, Jamshed Iqbal
Topics & Concepts
ChemistryMonoamine oxidaseCholinesteraseIn silicoIn vitroMonoamine neurotransmitterPharmacologyMonoamine oxidase BBiochemistryEnzymeCombinatorial chemistrySerotoninReceptorMedicineGeneCholinesterase and Neurodegenerative DiseasesNicotinic Acetylcholine Receptors StudySynthesis and biological activity