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A potential cocrystal strategy to tailor in-vitro dissolution and improve Caco-2 permeability and oral bioavailability of berberine

Hui Chen, Jiangpo Ma, Feng Zhou, Junhui Yang, Lei Jiang, Quanbing Chen, Yang Zhou, Jiantao Zhang, Jiantao Zhang

2024International Journal of Pharmaceutics12 citationsDOI

Topics & Concepts

CocrystalBioavailabilityBerberineCaco-2DissolutionChemistryPermeability (electromagnetism)PharmacologyIn vitroBiochemistryMedicineOrganic chemistryMembraneMoleculeHydrogen bondBerberine and alkaloids researchAlkaloids: synthesis and pharmacologyChemical synthesis and alkaloids
A potential cocrystal strategy to tailor in-vitro dissolution and improve Caco-2 permeability and oral bioavailability of berberine | Litcius