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Design, synthesis and biological evaluations of a long-acting, hypoxia-activated prodrug of fasudil, a ROCK inhibitor, to reduce its systemic side-effects

Taslim A. Al‐Hilal, Mohammad Anwar Hossain, Ahmed Alobaida, Farzana Alam, Ali Keshavarz, Eva Nozik‐Grayck, Kurt R. Stenmark, Nadezhda German, Fakhrul Ahsan

2021Journal of Controlled Release36 citationsDOIOpen Access PDF

Topics & Concepts

FasudilProdrugHypoxia (environmental)PharmacologyRho kinase inhibitorChemistryRho-associated protein kinaseMedicineBiochemistryKinaseOxygenOrganic chemistryCancer, Hypoxia, and MetabolismProtein Kinase Regulation and GTPase SignalingNitric Oxide and Endothelin Effects
Design, synthesis and biological evaluations of a long-acting, hypoxia-activated prodrug of fasudil, a ROCK inhibitor, to reduce its systemic side-effects | Litcius