Human PLD structures enable drug design and characterization of isoenzyme selectivity
Claire M. Metrick, Emily A. Peterson, Joseph C. Santoro, Istvan Enyedy, Paramasivam Murugan, TeYu Chen, Klaus Michelsen, Michael L. Cullivan, Kerri Spilker, P. Rajesh Kumar, Tricia L. May‐Dracka, Jayanth V. Chodaparambil
Topics & Concepts
IsozymeEnzymePhosphatidic acidPhospholipase DBiochemistryGene isoformBiologyDrug discoveryHomology modelingChemistryComputational biologyGeneMembranePhospholipidCholinesterase and Neurodegenerative DiseasesPhosphodiesterase function and regulationEnzyme function and inhibition