Design and synthesis of quinoline-pyrimidine inspired hybrids as potential plasmodial inhibitors
Francis Kayamba, Teboho Malimabe, Idowu Kehinde Ademola, Ofentse Jacob Pooe, Narva Deshwar Kushwaha, Mavela Cleopus Mahlalela, Robyn L. van Zyl, Michelle Gordon, Pertunia T. Mudau, Tawanda Zininga, Addmore Shonhai, Vincent O. Nyamori, Rajshekhar Karpoormath
Topics & Concepts
ChemistryPlasmodium falciparumPyrimidineDocking (animal)IC50StereochemistryCombination therapyArtemisininPharmacologyIn vitroBiochemistryMalariaBiologyMedicineImmunologyNursingMalaria Research and ControlComputational Drug Discovery MethodsResearch on Leishmaniasis Studies