Ligand recognition and allosteric regulation of DRD1-Gs signaling complexes
Peng Xiao, Wei Yan, Lu Gou, Ya-Ni Zhong, Liangliang Kong, Chao Wu, Xin Wen, Yuan Yuan, Sheng Cao, Changxiu Qu, Xin Yang, Chuan-Cheng Yang, Anjie Xia, Zhenquan Hu, Qianqian Zhang, Yong He, Daolai Zhang, Chao Zhang, Gui-Hua Hou, Huanxiang Liu, Lizhe Zhu, Ping Fu, Shengyong Yang, Daniel M. Rosenbaum, Jin‐Peng Sun, Yang Du, Lei Zhang, Xiao Yu, Zhenhua Shao
Topics & Concepts
Allosteric regulationBiologyDopamineDopamine receptorAgonistReceptorEndogenous agonistBinding siteLigand (biochemistry)Dopamine receptor D1Allosteric enzymeDopamine receptor D2G protein-coupled receptorAllosteric modulatorCell biologyBiophysicsNeuroscienceBiochemistryReceptor Mechanisms and SignalingProtein Structure and DynamicsComputational Drug Discovery Methods