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KI‐Mediated One‐Pot Transition‐Metal‐Rree Synthesis of 4‐Phenylpyrrolo[1,2‐<i>a</i>]quinoxalines

Shichen Li, Caixia Xie, Xianglong Chu, Zhen Dai, Lei Feng, Chen Ma

2020European Journal of Organic Chemistry22 citationsDOI

Abstract

An efficient and eco‐friendly method for the synthesis of pyrrolo[1,2‐ a ]quinoxalines is presented. Compared to previous methods, this protocol is transition‐metal‐free and only potassium iodide is required. A series of substituted 4‐phenylpyrrolo[1,2‐ a ]quinoxalines are obtained in moderate to good yields.

Topics & Concepts

ChemistryTransition metalCombinatorial chemistryEnvironmentally friendlyPotassiumIodineOrganic chemistryCatalysisEcologyBiologySynthesis and Biological EvaluationSynthesis and Characterization of PyrrolesMulticomponent Synthesis of Heterocycles