Discovery and optimization of novel pyrazole-benzimidazole CPL304110, as a potent and selective inhibitor of fibroblast growth factor receptors FGFR (1–3)
Abdellah Yamani, Daria Zdżalik-Bielecka, Joanna Lipner, Aleksandra Stańczak, Natalia Piórkowska, Paulina Seweryna Stańczak, Patrycja Olejkowska, Joanna Hucz‐Kalitowska, Marta Magdycz, Karolina Dzwonek, Krzysztof Dubiel, Monika Lamparska‐Przybysz, Delfina Popiel, Jerzy Pieczykolan, Maciej Wieczorek
Topics & Concepts
ChemistryFibroblast growth factor receptorBenzimidazolePyrazoleReceptorFibroblast growth factorFibroblast growth factor receptor 3Fibroblast growth factor receptor 1Combinatorial chemistryBiochemistryPharmacologyStereochemistryOrganic chemistryMedicineFibroblast Growth Factor ResearchKruppel-like factors researchEosinophilic Disorders and Syndromes