Litcius/Paper detail

Recent progress in topoisomerase inhibitors as anticancer agents: Research and design strategies for Topo I and II inhibitors via structural optimization

G. D. Shen, Shihao Li, Yu Zhu, Zheng Xu, Xuan Liu, Chen Lv, Zhihua Xing, Linlin Cui, Wenlan Li

2025Bioorganic Chemistry11 citationsDOI

Topics & Concepts

TopoisomeraseTopoisomerase inhibitorChemistryEnzymeComputational biologyDNACancerCancer cellCell growthPharmacologyBiochemistryCancer researchEnzyme inhibitorCancer therapyDrugDNA damageBiologyDrug discoveryTumor cellsCancer therapeutics and mechanismsSynthesis and biological activityBioactive Compounds and Antitumor Agents