Metabolism-guided development of Ko143 analogs as ABCG2 inhibitors
Junjie Zhu, Saifei Lei, Jie Lu, Yixuan Hao, Qian Qi, Aaron S. Devanathan, Zhiwei Feng, Xiang‐Qun Xie, Peter Wipf, Xiaochao Ma
Topics & Concepts
ChemistryAbcg2MoietyAmideEffluxPharmacologySubfamilyBiochemistryTransporterStereochemistryATP-binding cassette transporterBiologyGeneDrug Transport and Resistance MechanismsCholesterol and Lipid MetabolismPharmacogenetics and Drug Metabolism