Litcius/Paper detail

2-Anilinoquinoline based arylamides as broad spectrum anticancer agents with B-RAFV600E/C-RAF kinase inhibitory effects: Design, synthesis, in vitro cell-based and oncogenic kinase assessments

Ashraf K. El‐Damasy, Md. Mamunul Haque, Jung Woo Park, Sang Chul Shin, Jun‐Seok Lee, Eunice EunKyeong Kim, Gyochang Keum

2020European Journal of Medicinal Chemistry24 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryKinaseBroad spectrumIn vitroPotencyIC50PharmacologyCancer cellApoptosisCancerCancer researchBiochemistryBiologyMedicineCombinatorial chemistryInternal medicineCancer Mechanisms and TherapyMelanoma and MAPK PathwaysChronic Myeloid Leukemia Treatments