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Discovery of novel non-steroidal selective glucocorticoid receptor modulators by structure- and IGN-based virtual screening, structural optimization, and biological evaluation

Xueping Hu, Jinping Pang, Changwei Chen, Dejun Jiang, Chao Shen, Xin Chai, Yang Liu, Xujun Zhang, Lei Xu, Sunliang Cui, Tingjun Hou, Dan Li

2022European Journal of Medicinal Chemistry26 citationsDOIOpen Access PDF

Topics & Concepts

TransrepressionTransactivationVirtual screeningGlucocorticoid receptorChemistryDocking (animal)IC50ReceptorPharmacologyIn silicoTranscription factorDrug discoveryBiochemistryMedicineIn vitroGeneNursingEstrogen and related hormone effectsCytokine Signaling Pathways and InteractionsVitamin D Research Studies
Discovery of novel non-steroidal selective glucocorticoid receptor modulators by structure- and IGN-based virtual screening, structural optimization, and biological evaluation | Litcius