Litcius/Paper detail

PROTACs to address the challenges facing small molecule inhibitors

Pedro Martín-Acosta, Xiangshu Xiao

2020European Journal of Medicinal Chemistry162 citationsDOIOpen Access PDF

Topics & Concepts

Drug discoverySmall moleculeAllosteric regulationChemistryUbiquitin ligaseChemical biologyComputational biologyLinkerProtein degradationUbiquitinNanotechnologyBiochemistryBiologyComputer scienceReceptorGeneOperating systemMaterials scienceProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments