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OligoTRAFTACs: A generalizable method for transcription factor degradation

Kusal T. G. Samarasinghe, Elvira An, Miriam A. Genuth, Ling Chu, Scott A. Holley, Craig M. Crews

2022RSC Chemical Biology50 citationsDOIOpen Access PDF

Abstract

Targeted transcription factor degradation using oligonucleotide-based transcription factor targeting chimeras (TRAFTACs).

Topics & Concepts

BrachyuryTranscription factorComputational biologyBiologyZebrafishUbiquitin ligaseCell biologyGeneGeneticsUbiquitinEmbryonic stem cellMesodermProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysGenomics and Chromatin Dynamics
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