Litcius/Paper detail

ARAF mutations confer resistance to the RAF inhibitor belvarafenib in melanoma

Ivana Yen, Frances Shanahan, Jeeyun Lee, Yong Sang Hong, Sang Joon Shin, Amanda R. Moore, Jawahar Sudhamsu, Matthew T. Chang, InHwan Bae, Darlene Dela Cruz, Thomas Hunsaker, Christiaan Klijn, Nicholas P. D. Liau, Eva Lin, Scott E. Martin, Zora Modrušan, Robert Piskol, Ehud Segal, Avinashnarayan Venkatanarayan, Xin Ye, Jianping Yin, Liangxuan Zhang, Jin-Soo Kim, Hyeong-Seok Lim, Kyu-pyo Kim, Yu Jung Kim, Hye Sook Han, Soo Jung Lee, Seung Tae Kim, Minkyu Jung, Yoon-Hee Hong, Young Su Noh, Munjeong Choi, Oakpil Han, Małgorzata Nowicka, Shrividhya Srinivasan, Yibing Yan, Tae Won Kim, Shiva Malek

2021Nature135 citationsDOIOpen Access PDF

Topics & Concepts

Neuroblastoma RAS viral oncogene homologMutantMelanomaMutationMEK inhibitorCancer researchKinasePharmacologyMedicineBiologyGeneticsMAPK/ERK pathwayGeneKRASMelanoma and MAPK PathwaysComputational Drug Discovery MethodsCancer Mechanisms and Therapy