The synthetic oleanane triterpenoid CDDO-Me binds and inhibits pyruvate kinase M2
Iaci N. Soares, Raiane Viana, Charles B. Trelford, Eddie Chan, Boun Thai, Elio A. Cino, Gianni M. Di Guglielmo
Topics & Concepts
PKM2Pyruvate kinaseChemistryWarburg effectGene knockdownCell cultureCell migrationCell biologyBiochemistryGlycolysisCellBiologyEnzymeApoptosisGeneticsCancer, Hypoxia, and MetabolismGlycosylation and Glycoproteins ResearchATP Synthase and ATPases Research