TRPV1 analgesics disturb core body temperature via a biased allosteric mechanism involving conformations distinct from that for nociception
Yizhe Huang, Jiating Ma, Yu-Jing Bian, Qin-Ru Bai, Yuhao Gao, S. Di, Yuntao Lei, Hui Yang, Xiaona Yang, Chang-Yan Shao, Wenhui Wang, Peng Cao, Changzhu Li, Michael X. Zhu, Mengyang Sun, Ye Yu
Topics & Concepts
NociceptionAllosteric regulationMechanism (biology)TRPV1Core (optical fiber)NeuroscienceChemistryPsychologyBiophysicsComputer scienceBiologyReceptorTransient receptor potential channelPhysicsBiochemistryTelecommunicationsQuantum mechanicsIon Channels and ReceptorsPain Mechanisms and TreatmentsNeurobiology and Insect Physiology Research