Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Nikolai Y. Zyk, Anton P. Ber, Ekaterina A. Nimenko, Radik R. Shafikov, Sergei Evteev, Stanislav A. Petrov, Anastasia A. Uspenskaya, Natalia Dashkova, Yan A. Ivanenkov, Dmitry A. Skvortsov, Елена К. Белоглазкина, Alexander G. Majouga, Aleksei E. Machulkin
Topics & Concepts
ChemistryMoietyLysineSelectivityNitrogen atomCombinatorial chemistryIn vitroConjugateStereochemistryBiochemistryOrganic chemistryAmino acidAlkylCatalysisMathematicsMathematical analysisProstate Cancer Treatment and ResearchRadiopharmaceutical Chemistry and ApplicationsMass Spectrometry Techniques and Applications