Discovery of pimozide derivatives as novel T-type calcium channel inhibitors with little binding affinity to dopamine D2 receptors for treatment of somatic and visceral pain
Yoshihito Kasanami, Chihiro Ishikawa, Takahiro Kino, Momoka Chonan, Naoki Toyooka, Yasuhiro Takashima, Yuriko Iba, Fumiko Sekiguchi, Maho Tsubota, Tsuyako Ohkubo, S. Yoshida, Atsushi Kawase, Takuya Okada, Atsufumi Kawabata
Topics & Concepts
PimozideChemistryDopamine receptor D2CatalepsyPharmacologyDopamineReceptorDopamine receptorCalcium channelNeuroscienceHaloperidolMedicineBiochemistryCalciumPsychologyOrganic chemistryIon channel regulation and functionPain Mechanisms and TreatmentsPharmacological Receptor Mechanisms and Effects