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Discovery of pimozide derivatives as novel T-type calcium channel inhibitors with little binding affinity to dopamine D2 receptors for treatment of somatic and visceral pain

Yoshihito Kasanami, Chihiro Ishikawa, Takahiro Kino, Momoka Chonan, Naoki Toyooka, Yasuhiro Takashima, Yuriko Iba, Fumiko Sekiguchi, Maho Tsubota, Tsuyako Ohkubo, S. Yoshida, Atsushi Kawase, Takuya Okada, Atsufumi Kawabata

2022European Journal of Medicinal Chemistry13 citationsDOIOpen Access PDF

Topics & Concepts

PimozideChemistryDopamine receptor D2CatalepsyPharmacologyDopamineReceptorDopamine receptorCalcium channelNeuroscienceHaloperidolMedicineBiochemistryCalciumPsychologyOrganic chemistryIon channel regulation and functionPain Mechanisms and TreatmentsPharmacological Receptor Mechanisms and Effects
Discovery of pimozide derivatives as novel T-type calcium channel inhibitors with little binding affinity to dopamine D2 receptors for treatment of somatic and visceral pain | Litcius