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A comprehensive review of emerging approaches in machine learning for <i>de novo</i> PROTAC design

Yossra Gharbi, Rocío Mercado

2024Digital Discovery21 citationsDOIOpen Access PDF

Abstract

Machine learning (ML) accelerates PROTAC design by optimizing linkers and protein–ligase interactions, enabling selective protein degradation for therapeutic applications, particularly targeting previously undruggable proteins.

Topics & Concepts

Computer scienceArtificial intelligenceMachine learningAdvancements in Semiconductor Devices and Circuit DesignIntegrated Circuits and Semiconductor Failure AnalysisProtein Degradation and Inhibitors
A comprehensive review of emerging approaches in machine learning for <i>de novo</i> PROTAC design | Litcius