Inhibitory effects of organophosphate esters on carboxylesterase activity of rat liver microsomes
Yukie Tsugoshi, Yoko Watanabe, Yuka Tanikawa, Chika Inoue, Kazumi Sugihara, Hiroyuki Kojima, Shigeyuki Kitamura
Topics & Concepts
Triphenyl phosphateCarboxylesteraseTrisPhosphateChemistryOrganophosphateCarbamoyl phosphate synthetaseMicrosomeIC50StereochemistryMedicinal chemistryBiochemistryEnzymeIn vitroOrganic chemistryFire retardantBiologyPesticideAgronomyCholinesterase and Neurodegenerative DiseasesPesticide Exposure and ToxicityComputational Drug Discovery Methods