Discovery of novel hybrid tryptamine-rivastigmine molecules as potent AChE and BChE inhibitors exhibiting multifunctional properties for the management of Alzheimer's disease
Gauri Shankar, Prabhat Kumar, Sanskriti Rai, Aparajita Ghosh, Tanmaykumar Varma, Mushtaq Ahmad Wani, Sunil Kumar, Upesh Mandloi, Gireesh Kumar Singh, Prabha Garg, Onkar P. Kulkarni, Saripella Srikrishna, Saroj Kumar, Gyan Modi
Topics & Concepts
RivastigmineChemistryTryptamineAchéAcetylcholinesteraseButyrylcholinesteraseTacrineCholinesteraseGalantaminePharmacologyDiseaseDonepezilEnzymeBiochemistryDementiaInternal medicineMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsChemical synthesis and alkaloids