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The importance of plasma protein and tissue binding in a drug discovery program to successfully deliver a preclinical candidate

Elizabeth Hann, Karine Malagu, Andrew J. Stott, Huw D. Vater

2022Progress in medicinal chemistry24 citationsDOI

Topics & Concepts

Drug discoveryDrugPharmacologyPlasma protein bindingComputational biologyDrug developmentPlasma concentrationDrug candidateBinding siteBiologyBioinformaticsBiochemistryProtein Interaction Studies and Fluorescence AnalysisProtein purification and stabilityDrug Transport and Resistance Mechanisms
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