New thiourea and benzamide derivatives of 2-aminothiazole as multi-target agents against Alzheimer's disease: Design, synthesis, and biological evaluation
Burcu Kılıç, Merve Bardakkaya, Rahşan Ilıkçı Sağkan, Fatma Aksakal, Shakila Shakila, Deniz S. Doğruer
Topics & Concepts
ChemistryBenzamideThioureaButyrylcholinesteraseCholinesteraseIC50CytotoxicityStereochemistryPharmacologyBiochemistryEnzymeAchéAcetylcholinesteraseOrganic chemistryIn vitroMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsFree Radicals and Antioxidants