Cholinesterases, α-glycosidase, and carbonic anhydrase inhibition properties of 1H-pyrazolo[1,2-b]phthalazine-5,10-dione derivatives: Synthetic analogues for the treatment of Alzheimer's disease and diabetes mellitus
Parham Taslımı, Kadir Turhan, Fikret Türkan, Halide Sedef Karaman, Zuhal Turgut, İlhami Gülçın
Topics & Concepts
ChemistryPhthalazineCarbonic anhydraseDiabetes mellitusCarbonic Anhydrase IEnzymeAcetylcholinesteraseStereochemistryBiochemistryCombinatorial chemistryOrganic chemistryEndocrinologyMedicineCholinesterase and Neurodegenerative DiseasesEnzyme function and inhibitionSynthesis and biological activity