Discovery of dual-active ethionamide boosters inhibiting the Mycobacterium tuberculosis ESX-1 secretion system
Raphael Gries, Jason Chhen, Edeltraud van Gumpel, Sebastian J. Theobald, Lindsay Sonnenkalb, Christian Utpatel, Fabian Metzen, Manuel Koch, Tobias Dallenga, Kamel Djaout, Alain R. Baulard, Michael Dal Molin, Jan Rybniker
Topics & Concepts
EthionamideMycobacterium tuberculosisVirulenceProdrugTuberculosisMicrobiologyAntimycobacterialSecretionDrug discoveryBiologyChemistryMedicineEthambutolPharmacologyGeneBiochemistryPathologyTuberculosis Research and EpidemiologyCancer therapeutics and mechanismsAntibiotic Resistance in Bacteria