Discovery of new pyrazole-4-carboxamide analogues as potential anticancer agents targeting dual aurora kinase A and B
Digambar Yevale, Nishith Teraiya, Twinkle Lalwani, Mayur Dalasaniya, Saumya Patel, Nandan Dixit, Chetan B. Sangani, Sujeet Kumar, N. V. L. Sirisha Mulukuri, Tao Huang, Yongtao Duan, Jie Zhang
Topics & Concepts
ChemistryPyrazoleCarboxamideAurora kinaseKinaseDual (grammatical number)Aurora A kinaseStereochemistryPharmacologyCombinatorial chemistryBiochemistryApoptosisCell cycleMedicineArtLiteratureMicrotubule and mitosis dynamicsCancer-related Molecular PathwaysUbiquitin and proteasome pathways