Insights into the molecular mechanism of triazolopyrimidinone derivatives effects on the modulation of α1β2γ2 subtype of GABAA receptor: An in silico approach
Zohreh Shafiee, Leila Karami, Mahmood Akbari, Elham Rezaee, Malik Maaza, Sayyed Abbas Tabatabai, Gilda Karimi
Topics & Concepts
ADMEGABAA receptorIn silicoMolecular dynamicsChemistryProtein subunitBenzodiazepineBinding siteReceptorDocking (animal)Molecular modelStereochemistryPharmacologyBiochemistryBiologyIn vitroComputational chemistryMedicineGeneNursingNeuroscience and Neuropharmacology ResearchPharmacological Receptor Mechanisms and EffectsTryptophan and brain disorders