COR758, a negative allosteric modulator of GABAB receptors
Alessandra Porcu, Rafaela Mostallino, Valeria Serra, Miriam Melis, Valeria Sogos, Sarah Beggiato, Luca Ferraro, Fabrizio Manetti, Beatrice Gianibbi, Bernhard Bettler, Federico Corelli, Claudia Mugnaini, M. Paola Castelli
Topics & Concepts
Allosteric regulationGABAB receptorAllosteric modulatorAgonistHEK 293 cellsGTP'Cell biologyChemistryG protein-coupled receptorReceptorBiophysicsBiochemistryBiologyEnzymeReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology ResearchNicotinic Acetylcholine Receptors Study