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Chemical inhibition of DPP9 sensitizes the CARD8 inflammasome in HIV-1-infected cells

Kolin M. Clark, Josh G. Kim, Qiankun Wang, Hongbo Gao, Rachel M. Presti, Liang Shan

2022Nature Chemical Biology47 citationsDOIOpen Access PDF

Topics & Concepts

InflammasomePyroptosisNucleoside Reverse Transcriptase InhibitorHuman immunodeficiency virus (HIV)IntracellularIn vitroProteaseChemistryProtease inhibitor (pharmacology)Reverse-transcriptase inhibitorVirologyReverse transcriptaseBiologyEnzymeBiochemistryRNAAntiretroviral therapyViral loadReceptorGeneInflammasome and immune disordersPneumocystis jirovecii pneumonia detection and treatmentToxoplasma gondii Research Studies
Chemical inhibition of DPP9 sensitizes the CARD8 inflammasome in HIV-1-infected cells | Litcius