New insights in the paradigm of upregulation of tumoral PSMA expression by androgen receptor blockade: Enzalutamide induces PSMA upregulation in castration-resistant prostate cancer even in patients having previously progressed on enzalutamide
Florian Rosar, Sebastian Dewes, Martin Ries, Andrea Schaefer, Fadi Khreish, Stephan Maus, H Bohnenberger, Johannes Linxweiler, Mark Bartholomä, Carsten‐Henning Ohlmann, Samer Ezziddin
Topics & Concepts
EnzalutamideProstate cancerMedicineAndrogen receptorUrologyInternal medicineDownregulation and upregulationBlockadeOncologyAntiandrogenRadioligandCancerReceptorChemistryBiochemistryGeneProstate Cancer Treatment and ResearchProstate Cancer Diagnosis and TreatmentRadiopharmaceutical Chemistry and Applications