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Discovery of a potent G-protein-coupled receptor 119 agonist for the treatment of type 2 diabetes

Suresh Pola, Shailesh R. Shah, Harikishore Pingali, Pandurang Zaware, Baban Thube, Pankaj Makadia, Hoshang Patel, Debdutta Bandyopadhyay, Akshyaya Rath, Suresh Giri, Jitendra H. Patel, Ramchandra Ranvir, Sugantha Sundar, Harilal Patel, Jeevan Kumar, Mukul R. Jain

2021Bioorganic & Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

AgonistChemistryGlycemicGlucose homeostasisIn vivoType 2 diabetesPharmacologyReceptorDiabetes mellitusPartial agonistInsulinPotencyIn vitroEndocrinologyBiochemistryInsulin resistanceMedicineBiologyBiotechnologyDiabetes Treatment and ManagementReceptor Mechanisms and SignalingPancreatic function and diabetes
Discovery of a potent G-protein-coupled receptor 119 agonist for the treatment of type 2 diabetes | Litcius