Medicinal chemistry strategies for the development of protein tyrosine phosphatase SHP2 inhibitors and PROTAC degraders
Kai Tang, Yao-Nan Jia, Bin Yu, Hong‐Min Liu
Topics & Concepts
Protein tyrosine phosphataseChemistryProto-oncogene tyrosine-protein kinase SrcPhosphataseDual-specificity phosphataseMAPK/ERK pathwayReceptor tyrosine kinaseBiochemistrySignal transductionPTPN11TyrosineComputational biologyCell biologyEnzymeGeneBiologyMutationKRASProtein Tyrosine PhosphatasesGalectins and Cancer BiologyPeptidase Inhibition and Analysis