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Design and synthesis of pyrido[2,3-d]pyrimidine derivatives for a novel PAC1 receptor antagonist

Ichiro Takasaki, Ai Watanabe, Takuya Okada, Daisuke Kanayama, Ryota Nagashima, Miyu Shudo, Ayaka Shimodaira, Kazuto Nunomura, Bangzhong Lin, Yurie Watanabe, Hiroaki Gouda, Atsuro Miyata, Takashi Kurihara, Naoki Toyooka

2022European Journal of Medicinal Chemistry15 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPyrimidineAntagonistAnalgesicPharmacologyReceptor antagonistReceptorStereochemistryAllodyniaPharmacokineticsNeuropathic painHyperalgesiaBiochemistryNociceptionMedicineNeuropeptides and Animal PhysiologyPain Mechanisms and TreatmentsReceptor Mechanisms and Signaling
Design and synthesis of pyrido[2,3-d]pyrimidine derivatives for a novel PAC1 receptor antagonist | Litcius